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R
D G Cooper Patents in Chronological Order
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| 1. |
Transformation
of a penicillin sulfoxide ester to a cephalosporin antibiotic.
R. D. G. Cooper, France 1,561,048 (March 21, 1969). |
| 2. |
Conversion
of a penicillin sulfoxide ester to a cephalosporin antibiotic.
R. D. G. Cooper, South Africa 6,802, 780 (October 30, 1969). |
| 3. |
Oxidation
of cephalosporins to cephalosporin S-oxides. R. D. G. Cooper,
German Offen. 1,937,016 (April 9, 1970). |
| 4. |
Reduction
of D3- cephalosporin S-oxide. R. D. G. Cooper, G. V. Kaiser,
C. F. Murphy, E. M. Van Heyningen, J. A. Webber, and I. G.
Wright, German Offen. 1,940,080 (September 17, 1970). |
| 5. |
Antibiotic
2-acyloxycephalosporin, and intermediates. R. D. G. Cooper,
German Offen, 1,950,390 (October 1, 1970). |
| 6. |
2,6-Dizaz-4-thiabicyclo[3.2.0]hept-2-en-7-ones.
R. D. G. Cooper, German Offen. 2,029,099 (January 28, 1971). |
| 7. |
4-(N-Alkenylcarbamyl)
thiazoles. R. D. G. Cooper, U.S. 3,594,389 (July 20, 1971). |
| 8. |
Thiazolinoazetidinones.
R. D. G. Cooper and D. S. Fukuda, U.S. 3,681,380 (August 1,
1972). |
| 9. |
Azeto
[3,2-]thiazoles. , . R.D. G. Cooper German Offen. 2,205,144
(October 19, 1972). |
| 10. |
Cephalosporin
antibiotics. R. D. G. Cooper, German Offen. 2,457,851 (June
12, 1975). |
| 11. |
Ureido-substituted
cephalosporins. R. D. G. Cooper and D. K. Herron, German Offen.
2,514,019 (October 2, 1975). |
| 12. |
Acylureidocephalosporins.
R. D. G. Cooper and D. K. Herron, German Offen. 2,514,020
(October 2, 1975). |
| 13. |
Antibiotic
ureidocephalosporins. R. D. G. Cooper and D. K. Herron, France
2,265,394 (October 24, 1975). |
| 14. |
Hydroxy-substituted
phenylglycylamido-3-heterocyclic thiomethyl cephalosporins,
R. D. G. Cooper, U.S. 3,946,003 (March 23, 1976). |
| 15. |
7-(a-Furoylureidoaryl
and cyclohexadienylacetamido) cephalosporin antibiotics. R.
D. G. Cooper, U.S. 3,956,292 (May 11, 1976). |
| 16. |
7-[a-(Guanyl-l-ureido)
phenylacetamido]-3-substituted cephalosporin antibiotics.
R. D. G. Cooper, U.S. 4,039,535 (August 2, 1977). |
| 17. |
2-(Carbalkoxyethylsulfinyl)-3-oxo-a-isopropenylazetidineacetic
acids. R. D. G. Cooper, German Offen. 2,707,815 (September
1, 1977). |
| 18. |
4-(Formylthio)azetidin-2-ones
and ozonization process for them. R. D. G. Cooper and D. O.
Spry, U.S. 4,048,157 (September 13, 1977). |
| 19. |
Substituted
4-oxa-2,6-diazabicycloheptene compounds. R. D. G. Cooper,
G. A. Koppel, L. J. McShane, German Offen. 2,809,528 (September
14, 1978). |
| 20. |
2-Azetidinone
derivatives. R. D. G. Cooper, G. A. Koppel, and L. J. McShane,
German Offen. 2,809,529 (September 14, 1978). |
| 21. |
Chlorination
of thiazoline-azetidinones. R. D. G. Cooper, U.S. 4,430,268
(1984). |
| 22. |
Allylic
chlorination process and compounds prepared thereby. R. D.
G. Cooper, USP 4,578,531 (May 21, 1985). |
| 23. |
Benzothienylglycyl
cephalosporin derivatives. R. D. G. Cooper, B. J. Graves and
E. R. Lavagnino, USP 4,482,553 (November 13, 1984). |
| 24. |
Napthylglycyl
cephalosporin derivatives. L. C. Blaszczak, R. D. G. Cooper
and J. R. Turner, USP 4,490,370 (January, 1985). |
| 25. |
Preparation
of oxazalines. R. D. G. Cooper, J. M. Morin and L. R. Peters,
USP 4,587,053 (May 6, 1986). |
| 26. |
Chiral
synthesis of azetidinones. R. D. G. Cooper, USP 4,734,498
(1987). |
| 27. |
3ß-(3,4-Disubstituted
succininido) azetidinones and their preparation, useful as
intermediates for ß-lactam antibacterials. R. D. G.
Cooper, E. P. 252,744 (January 13, 1988). |
| 28. |
Chiral
azetidinones, useful as intermediates for the preparation
of ß-lactam antibiotics, and a procedure for their preparation.
R. D. G. Cooper, E. P. 254,578 (January 27, 1988). |
| 29. |
Preparation
and formulation of 7-Phenylglycyl-1-carba-1-dethiacephalosporins
as antibiotics. R. D. G. Cooper and J. W. Webber, E. P. 266,296
(May 11, 1988). |
| 30. |
Combinatorial
Process for Synthesizing Azetidinone Analogues. R.D.G.Cooper
et al. U.S. 5759865 (Feb. 6, 1998). |
| 31. |
New
Glycopeptide Derivatives. R.D.G.Cooper et al. E.P. 0667353
(Aug. 16 1995). |
| 32. |
Non-Peptidyl
Vasopressin V1a Derivatives. R.D.G.Cooper et al. WO 9730707A1,
(Aug. 28, 1997). |
| 33. |
Glycopeptide
Antibiotic Derivatives. R.D.G.Cooper et al. U.S. 584068 (Nov.
24, 1998). |
| 34. |
Glycopeptide
Amides. R.D.G.Cooper et al. W.O. 9800153A1 ( Jan. 8, 1998). |
| 35. |
Glycopeptide
Deacylation Process and Product. R.D.G.Cooper et al. WO 9846580A1,
( Oct. 22, 1998). |
| 36. |
Teichoplanin
Derivatives. R.D.G.Cooper et al. WO 9846579A1 ( Oct. 22, 1998) |
| 37. |
Glycopeptide
Antibiotic Derivatives. R.D.G.Cooper et al. U.S. 5843889 (Dec.
1, 1998). |
| 38. |
Glycopeptide
Amides. R.D.G. Cooper et al. U.S. 5,919,756 (July 6th. 1999). |
| 39. |
Glycopeptide
Antibiotic Derivatives. R.D.G. Cooper et al. U.S. 5,977,062
(Nov. 2, 1999). |
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